2412461-98-2

2412461-98-2 structure

2412461-98-2 structure

Name: UR-MB108
Chemical Name: UR-MB108
CAS Number: 2412461-98-2
Molecular Formula: C₄₀H₃₈N₆O₄
Molecular Weight: 666.77
Catalog: Signaling Pathways Membrane Transporter/Ion Channel BCRP
Create Date: 2022-07-01 17:14:31
Modify Date: 2024-02-03 20:45:39
UR-MB108 (Compound 57) is a potent, selective ABCG2 (BCRP) inhibitor with an IC50 of 79 nM. UR-MB108 is stable in blood plasma[1].

Name	UR-MB108

Description	UR-MB108 (Compound 57) is a potent, selective ABCG2 (BCRP) inhibitor with an IC50 of 79 nM. UR-MB108 is stable in blood plasma[1].
Related Catalog	Research Areas >> Cancer Signaling Pathways >> Membrane Transporter/Ion Channel >> BCRP
Target	IC50: 79 nM (ABCG2 (BCRP))[1]
References	[1]. Frauke Antoni, et al. Tariquidar-related triazoles as potent, selective and stable inhibitors of ABCG2 (BCRP). Eur J Med Chem. 2020 Apr 1;191:112133.

Molecular Formula	C₄₀H₃₈N₆O₄
Molecular Weight	666.77