2748687-95-6
2748687-95-6 structure
- Name: GSK737
- Chemical Name: GSK737
- CAS Number: 2748687-95-6
- Molecular Formula: C20H21N5O2
- Molecular Weight: 363.421
- Catalog: Signaling Pathways Epigenetics Epigenetic Reader Domain
- Create Date: 2022-07-13 12:56:43
- Modify Date: 2024-04-11 15:49:09
-
GSK737 (GSK-737) is a potent, highly selective BET BD2 inhibitor with pIC50 of 7.3 (BRD4 BD2), 200-fold selectivity over BRD4 BD1.
| Name | GSK737 |
|---|
| Description | GSK737 (GSK-737) is a potent, highly selective BET BD2 inhibitor with pIC50 of 7.3 (BRD4 BD2), 200-fold selectivity over BRD4 BD1. |
|---|---|
| References | 1. Helen E Aylott, et al. J Med Chem. 2021 Mar 25;64(6):3249-3281. |
| Molecular Formula | C20H21N5O2 |
|---|---|
| Molecular Weight | 363.421 |