2359618-49-6

2359618-49-6 structure

Name: BPTF-IN-1
Chemical Name: BPTF-IN-1
CAS Number: 2359618-49-6
Molecular Formula: C₂₃H₂₃FN₆O₃
Molecular Weight: 450.47
Catalog: Signaling Pathways Epigenetics Epigenetic Reader Domain
Create Date: 2022-07-12 11:36:49
Modify Date: 2025-08-25 18:27:47
BPTF-IN-1 (compound AU1) is a selective bromodomain and PHD finger containing transcription factor (BPTF) bromodomain inhibitor with a Kd of 2.8 μM. BPTF-IN-1 shows to be selective for BPTF over BRD4 bromodomain. BPTF-IN-1 shows antimalarial activity[1].

Name	BPTF-IN-1

Description	BPTF-IN-1 (compound AU1) is a selective bromodomain and PHD finger containing transcription factor (BPTF) bromodomain inhibitor with a Kd of 2.8 μM. BPTF-IN-1 shows to be selective for BPTF over BRD4 bromodomain. BPTF-IN-1 shows antimalarial activity[1].
Related Catalog	Research Areas >> Infection Signaling Pathways >> Epigenetics >> Epigenetic Reader Domain
References	[1]. Steven E Kirberger, et al. Selectivity, ligand deconstruction, and cellular activity analysis of a BPTF bromodomain inhibitor. Org Biomol Chem. 2019 Feb 13;17(7):2020-2027.

Molecular Formula	C₂₃H₂₃FN₆O₃
Molecular Weight	450.47