2166320-76-7
2166320-76-7 structure
- Name: Feniralstat
- Chemical Name: Feniralstat
- CAS Number: 2166320-76-7
- Molecular Formula: C26H25F2N5O4
- Molecular Weight: 509.50
- Catalog: Research Areas Cardiovascular Disease
- Create Date: 2022-04-06 04:39:46
- Modify Date: 2024-01-23 10:19:44
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Feniralstat (compound 30), a pyrazole derivative, is a potent kallikrein inhibitor with an IC50 of 6.7 nM for Human plasma kallikrein (pKal). Feniralstat has no inhibition on Human KLKl, Human FXIa, Human Factor Xlla (all IC50>40 μM).
| Name | Feniralstat |
|---|
| Description | Feniralstat (compound 30), a pyrazole derivative, is a potent kallikrein inhibitor with an IC50 of 6.7 nM for Human plasma kallikrein (pKal). Feniralstat has no inhibition on Human KLKl, Human FXIa, Human Factor Xlla (all IC50>40 μM). |
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| Related Catalog | |
| References |
[1]. Rebecca Louise DAVIE, et al. Pyrazole derivatives as plasma kallikrein inhibitors. WO2017207983A1. |
| Molecular Formula | C26H25F2N5O4 |
|---|---|
| Molecular Weight | 509.50 |