2009052-76-8
2009052-76-8 structure
- Name: VU 6001966
- Chemical Name: VU 6001966
- CAS Number: 2009052-76-8
- Molecular Formula: C17H15FN4O2
- Molecular Weight: 326.331
- Catalog: Signaling Pathways GPCR/G Protein mGluR
- Create Date: 2020-01-20 12:11:57
- Modify Date: 2024-09-29 12:34:08
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A potent and selective, CNS penetrant mGlu2 negative allosteric modulator with IC50 of 78 nM; shows no inhibition for mGlu3 (IC50>30 uM); represents an exciting lead series for potential mGlu2 PET tracer development.
| Name | VU 6001966 |
|---|
| Description | A potent and selective, CNS penetrant mGlu2 negative allosteric modulator with IC50 of 78 nM; shows no inhibition for mGlu3 (IC50>30 uM); represents an exciting lead series for potential mGlu2 PET tracer development. |
|---|---|
| References | References 1. Bollinger KA, et al. ACS Med Chem Lett. 2017 Aug 3;8(9):919-924. View Related Products by Target mGluR |
| Molecular Formula | C17H15FN4O2 |
|---|---|
| Molecular Weight | 326.331 |