2101206-81-7
2101206-81-7 structure
- Name: CAM4066
- Chemical Name: N-[(2-Chloro-4-biphenylyl)methyl]-β-alanyl-N-(3-carboxyphenyl)-β-alaninamide
- CAS Number: 2101206-81-7
- Molecular Formula: C26H26ClN3O4
- Molecular Weight: 479.955
- Create Date: 2020-01-11 17:35:58
- Modify Date: 2023-01-20 08:48:13
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CAM4066 (CAM-4066) is a potent and selective CK2α inhibitor with Kd of 0.32 uM and IC50 of 0.37 uM, shows significantly improved selectivity compared to other CK2α inhibitors.
| Name | N-[(2-Chloro-4-biphenylyl)methyl]-β-alanyl-N-(3-carboxyphenyl)-β-alaninamide |
|---|---|
| Synonyms |
N-[(2-Chloro-4-biphenylyl)methyl]-β-alanyl-N-(3-carboxyphenyl)-β-alaninamide
β-Alaninamide, N-[(2-chloro[1,1'-biphenyl]-4-yl)methyl]-β-alanyl-N-(3-carboxyphenyl)- N-[(2-Chlorobiphenyl-4-Yl)methyl]-β-Alanyl-N-(3-Carboxyphenyl)-β-Alaninamide |
| Description | CAM4066 (CAM-4066) is a potent and selective CK2α inhibitor with Kd of 0.32 uM and IC50 of 0.37 uM, shows significantly improved selectivity compared to other CK2α inhibitors. |
|---|---|
| References | References 1. Iegre J, et al. Chem Sci. 2018 Feb 20;9(11):3041-3049. 2. Brear P, et al. Chem Sci. 2016 Nov 1;7(11):6839-6845. 3. De Fusco C, et al. Bioorg Med Chem. 2017 Jul 1;25(13):3471-3482. View Related Products by Target Casein Kinase |
| Density | 1.3±0.1 g/cm3 |
|---|---|
| Boiling Point | 780.2±60.0 °C at 760 mmHg |
| Molecular Formula | C26H26ClN3O4 |
| Molecular Weight | 479.955 |
| Flash Point | 425.6±32.9 °C |
| Exact Mass | 479.161194 |
| LogP | 4.30 |
| Vapour Pressure | 0.0±2.8 mmHg at 25°C |
| Index of Refraction | 1.630 |