2130869-18-8

2130869-18-8 structure
2130869-18-8 structure
  • Name: Mal-PEG2-VCP-Eribulin
  • Chemical Name: Mal-PEG2-VCP-Eribulin
  • CAS Number: 2130869-18-8
  • Molecular Formula: C70H99N7O21
  • Molecular Weight: 1374.57
  • Catalog: Signaling Pathways Antibody-drug Conjugate Drug-Linker Conjugates for ADC
  • Create Date: 2019-09-07 12:13:18
  • Modify Date: 2025-08-23 03:20:57
  • Mal-PEG2-VCP-Eribulin consists the ADCs linker (Mal-PEG2-VCP) and Eribulin[1]. Eribulin is a mechanistically unique microtubule inhibitor for cancer[2]. Mal-PEG2-VCP-Eribulin is an Eribulin-based drug for antibody conjugates[1].

Name Mal-PEG2-VCP-Eribulin
Description Mal-PEG2-VCP-Eribulin consists the ADCs linker (Mal-PEG2-VCP) and Eribulin[1]. Eribulin is a mechanistically unique microtubule inhibitor for cancer[2]. Mal-PEG2-VCP-Eribulin is an Eribulin-based drug for antibody conjugates[1].
Related Catalog
References

[1]. Earl F Albone, et al. Eribulin-based antibody-drug conjugates and methods of use. US20170252458A1.

[2]. Towle MJ, et al. Eribulin induces irreversible mitotic blockade: implications of cell-based pharmacodynamics for in vivo efficacy under intermittent dosing conditions. Cancer Res. 2011 Jan 15;71(2):496-505.

Molecular Formula C70H99N7O21
Molecular Weight 1374.57
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