1883863-52-2
1883863-52-2 structure
- Name: dBET57
- Chemical Name: dBET57
- CAS Number: 1883863-52-2
- Molecular Formula: C34H31ClN8O5S
- Molecular Weight: 699.18
- Catalog: Signaling Pathways Epigenetics Epigenetic Reader Domain
- Create Date: 2019-08-04 09:55:58
- Modify Date: 2024-04-09 14:37:15
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dBET57 is a potent and selective heterobifunctional degrader of BRD4 based on the PROTAC technology, with a DC50/5h of 500 nM for BRD4BD1, and is inactive on BRD4BD2[1].
| Name | dBET57 |
|---|
| Description | dBET57 is a potent and selective heterobifunctional degrader of BRD4 based on the PROTAC technology, with a DC50/5h of 500 nM for BRD4BD1, and is inactive on BRD4BD2[1]. |
|---|---|
| Related Catalog | |
| Target |
DC50/5h: 500 nM (BRD4BD1)[1] |
| References |
| Molecular Formula | C34H31ClN8O5S |
|---|---|
| Molecular Weight | 699.18 |