Shanghai Nianxing Industrial Co., Ltd
China
Product Name: GSK3395879
Price: Check
Purity: 98.0%
Stocking Period: 10 Day
Contact: Yang
Email: sales@echemcloud.com

DC Chemicals Limited
China
Product Name: GSK3395879
Price: $Inquiry/100mg ￥Inquiry/250mg ￥Inquiry/1g
Purity: 98.0%
Stocking Period: Inquiry
Contact: Tony Cao
Email: sales@dcchemicals.com

2215852-91-6

2215852-91-6 structure

2215852-91-6 structure

Name: GSK3395879
Chemical Name: GSK3395879
CAS Number: 2215852-91-6
Molecular Formula: C₂₀H₁₅F₄N₃O₅S
Molecular Weight: 485.41
Catalog: Signaling Pathways Membrane Transporter/Ion Channel TRP Channel
Create Date: 2019-06-04 18:10:27
Modify Date: 2024-01-19 12:06:30
GSK3395879 is a selective and orally bioavailable transient receptor potential vanilloid-4 (TRPV4) antagonist with an IC50 of 1 nM for hTRPV4[1].

Name	GSK3395879

Description	GSK3395879 is a selective and orally bioavailable transient receptor potential vanilloid-4 (TRPV4) antagonist with an IC50 of 1 nM for hTRPV4[1].
Related Catalog	Signaling Pathways >> Membrane Transporter/Ion Channel >> TRP Channel Research Areas >> Cardiovascular Disease
Target	IC50: 1 nM (hTRPV4)[1]
References	[1]. Brnardic EJ, et al. Discovery of Pyrrolidine Sulfonamides as Selective and Orally Bioavailable Antagonists of Transient Receptor Potential Vanilloid-4 (TRPV4). J Med Chem. 2018 Nov 8;61(21):9738-9755.

Molecular Formula	C₂₀H₁₅F₄N₃O₅S
Molecular Weight	485.41

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