2230850-47-0

2230850-47-0 structure

Name: EHMT2-IN-2
Chemical Name: EHMT2-IN-2
CAS Number: 2230850-47-0
Molecular Formula: C₂₁H₂₂N₆O
Molecular Weight: 374.44
Catalog: Signaling Pathways Epigenetics Histone Methyltransferase
Create Date: 2019-06-02 09:59:08
Modify Date: 2025-09-18 23:01:21
EHMT2-IN-2 is a potent EHMT inhibitor, with IC50s of all <100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2. Used in the research of blood disease or cancer[1].

Name	EHMT2-IN-2

Description	EHMT2-IN-2 is a potent EHMT inhibitor, with IC50s of all <100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2. Used in the research of blood disease or cancer[1].
Related Catalog	Research Areas >> Cancer Signaling Pathways >> Epigenetics >> Histone Methyltransferase
Target	EHMTI PEP:<100 nM (IC50) EHMT2 PEP:<100 nM (IC50) EHMT2 ICW:<100 nM (IC50)
In Vitro	EHMT2-IN-2 (Compound 200) is a potent EHMT inhibitor, with IC50s of all < 100 nM for EEHMT1 peptide, EHMT2 peptide and cellular EHMT2[1].
References	[1]. John Emmerson Campbell, et al. Amine-substituted heterocyclic compounds as ehmt2 inhibitors and methods of use thereof. WO2018118842A1.