PEN-221

Names

[ CAS No. ]:
1853254-97-3

[ Name ]:
PEN-221

Biological Activity

[Description]:

PEN-221 is a Somatostatin receptor 2 (SSTR2)-targeting cytotoxic conjugate with an IC50 of 10 nM.

[Related Catalog]:

Research Areas >> Cancer

Signaling Pathways >> GPCR/G Protein >> Somatostatin Receptor

[Target]

IC50: 10 nM (SSTR2)[1]

[References]

[1]. White BH, et al. Discovery of an SSTR2-Targeting Maytansinoid Conjugate (PEN-221) with Potent Activity in Vitro and in Vivo. J Med Chem. 2019 Mar 14;62(5):2708-2719.

Chemical & Physical Properties

[ Molecular Formula ]:
C₈₃H₁₀₉ClN₁₄O₂₀S₄

[ Molecular Weight ]:
1786.55

Related Compounds

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