ACAT-IN-1 cis isomer

Names

[ CAS No. ]:
145961-79-1

[ Name ]:
ACAT-IN-1 cis isomer

Biological Activity

[Description]:

ACAT-IN-1 cis isomer is a potent ACAT inhibitor with an IC50 of 100 nM.

[Related Catalog]:

Signaling Pathways >> Metabolic Enzyme/Protease >> Acyltransferase
Research Areas >> Metabolic Disease

[Target]

IC50: 100 nM (ACAT)[1]


[References]

[1]. Vaccaro W, et al. Inhibitors of Acyl CoA:Cholesterol Acyltransferase. J. Med. Chem., 1996, 39 (8), pp 1704–1719


[Related Small Molecules]

Avasimibe | LCQ-908 | DGAT-3 | A922500 | Xanthohumol | PF-04620110 | AZD7687 | MGAT2-IN-1 | DGAT-1 inhibitor 2 | DGAT1-IN-1 | K-604 dihydrochloride | PF-06471553 | YM17E | ABT-046 | RP 70676

Chemical & Physical Properties

[ Molecular Formula ]:
C29H25NO2

[ Molecular Weight ]:
419.51


Related Compounds