5-HT3 antagonist 1

Names

[ CAS No. ]:
129294-09-3

[ Name ]:
5-HT3 antagonist 1

[Synonym ]:
(+/-)-N-[1-methyl-4-(3-methylbenzyl)hexahydro-1H-1,4-diazepin-6-yl]-1H-indazole-3-carboxamide
1H-Indazole-3-carboxylic acid [1-methyl-4-(3-methyl-benzyl)-[1,4]diazepan-6-yl]-amide
N-[1-methyl-4-(3-methylbenzyl)hexahydro-1H-1,4-diazepin-6-yl]-1H-indazole-3-carboxamide
5-HT3 antagonist 1

Biological Activity

[Description]:

5-HT3 antagonist 1 is a potent and selective antagonist of serotonin 3 (5-HT3) receptor.

[Related Catalog]:

Signaling Pathways >> GPCR/G Protein >> 5-HT Receptor
Signaling Pathways >> Neuronal Signaling >> 5-HT Receptor
Research Areas >> Neurological Disease

[References]

[1]. INDAZOLE-3-CARBOXYLIC ACID DERIVATIVES. US5017573


[Related Small Molecules]

Harmine | Pimavanserin | Serotonin hydrochloride | Sodium Ferulate | Thioridazine hydrochloride | Brexpiprazole | Risperidone | TG6-10-1 | Cariprazine | Quetiapine | SERTINDOLE | Alprenolol hydrochloride | B-HT 920 | Ketanserin | Palonosetron hydrochloride

Chemical & Physical Properties

[ Molecular Formula ]:
C22H27N5O

[ Molecular Weight ]:
377.48300

[ Exact Mass ]:
377.22200

[ PSA ]:
64.26000

[ LogP ]:
2.68400

Related Compounds