ALPK1-IN-2

Names

[ CAS No. ]:
2765633-68-7

[ Name ]:
ALPK1-IN-2

Biological Activity

[Description]:

ALPK1-IN-2 (compound T001) is a potent ALPK1 (alpha-kinase 1) inhibitor, with an IC50 of 95 nM. ALPK1-IN-2 also inhibits NF-κB, with an IC50 of 1.31 μM[1].

[Related Catalog]:

Research Areas >> Cancer
Research Areas >> Inflammation/Immunology

[Target]

IC50: 95 nM (ALPK1), 1.31 μM (NF-κB)[1]


[References]

[1]. Danyang Liu, et al. Benzothiazole and quinoline derivatives and their use. WO2022063153A1.

Chemical & Physical Properties

[ Molecular Formula ]:
C20H18F2N4O2S

[ Molecular Weight ]:
416.44

Related Compounds