CPI-0610 carboxylic acid

Names

[ CAS No. ]:
1380089-81-5

[ Name ]:
CPI-0610 carboxylic acid

Biological Activity

[Description]:

CPI-0610 carboxylic acid is a ligand for target protein for protact. CPI-0610 carboxylic acid is a potent bromodomain and extra-terminal (BET) protein inhibitor in the therapy of multiple myeloma[1].

[Related Catalog]:

Research Areas >> Cancer
Signaling Pathways >> Epigenetics >> Epigenetic Reader Domain

[Target]

BET[1]


[References]

[1]. Albrecht BK, et al. Identification of a Benzoisoxazoloazepine Inhibitor (CPI-0610) of the Bromodomain and Extra-Terminal (BET) Family as a Candidate for Human Clinical Trials. J Med Chem. 2016 Feb 25;59(4):1330-9.

Chemical & Physical Properties

[ Molecular Formula ]:
C20H15ClN2O3

[ Molecular Weight ]:
366.80

Related Compounds