NVP-BDZ 824
Names
[ CAS No. ]:
916306-04-2
[ Name ]:
NVP-BDZ 824
Biological Activity
[Description]:
A potent, highly selective antagonist of chemokine receptor CXCR3 with binding IC50 of 146 nM, Ca2+-mobilization IC50 of 28 nM.
[References]
References 1. Thoma G, et al. Bioorg Med Chem Lett. 2009 Nov 1;19(21):6185-8. 2. Bernat V, et al. ChemMedChem. 2012 Aug;7(8):1481-9. View Related Products by Target Chemokine Receptor (CCR and CXCR)
Chemical & Physical Properties
[ Molecular Formula ]:
C27H30N4O2
[ Molecular Weight ]:
442.563