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CPUY074020

Names

[ CAS No. ]:
902279-44-1

[ Name ]:
CPUY074020

[Synonym ]:
MFCD14777686

Biological Activity

[Description]:

CPUY074020 is a potent G9a inhibitor with an IC50 of 2.18 μM, and possesses anti-proliferative activity [1].

[Related Catalog]:

Research Areas >> Cancer

Signaling Pathways >> Epigenetics >> Histone Methyltransferase

[Target]

IC50: 2.18 μM (G9a)[1]

[References]

[1]. Chen WL, et al. Discovery, design and synthesis of 6H-anthra[1,9-cd]isoxazol-6-one scaffold as G9a inhibitor through a combination of shape-based virtual screening and structure-based molecular. Bioorg Med Chem. 2016 Nov 15;24(22):6102-6108.

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₅H₂₈N₄O₂

[ Molecular Weight ]:
416.52

Related Compounds