GPR132 antagonist 1

Names

[ Name ]:
GPR132 antagonist 1

Biological Activity

[Description]:

GPR132 antagonist 1 (GPR132-B-160, Compound 25) is a GPR132 antagonist with an EC50 value of 0.075 μM. GPR132 antagonist 1 has promote insulin secretion activity with an EC50 value of 0.7 μM[1].

[Related Catalog]:

Signaling Pathways >> Others >> Others

Research Areas >> Metabolic Disease

[Target]

EC50: 0.075 μM (GPR132); 0.7 μM (insulin secretion activity)[1].

[References]

[1]. 焦宁, 等. Gpcr调节剂及其应用. 专利. CN116903563A.

Chemical & Physical Properties

[ Molecular Formula ]:
C₁₈H₁₇NO₅S

[ Molecular Weight ]:
359.40

Related Compounds

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