WAY 207024 dihydrochloride

Names

[ CAS No. ]:
872002-73-8

[ Name ]:
WAY 207024 dihydrochloride

[Synonym ]:
6-[[4-[2-[4-(1,1-Dimethylethyl)phenyl]-1H-benzimidazol-7-yl]-i-piperazinyl]methyl]-quinoxalinedihydrochloride
2-(4-tert-Butylphenyl)-4-[4-[(6-quinoxalyl)methyl]piperazin-1-yl]benzimidazole dihydrochloride
WAY 207024 DIHYDROCHLORIDE
Quinoxaline, 6-[[4-[2-[4-(1,1-dimethylethyl)phenyl]-1H-benzimidazol-4-yl]-1-piperazinyl]methyl]-, dihydrochloride
WAY-207024 DIHYDROCHLORIDE
A 68930 hydrochloride

Biological Activity

[Description]:

WAY-207024 (dihydrochloride) is a potent and orally active GnRH antagonist that reduces leuteinizing hormone (LH) levels in plasma[1].

[Related Catalog]:

Signaling Pathways >> GPCR/G Protein >> GNRH Receptor

Research Areas >> Cardiovascular Disease

[References]

[1]. Pelletier JC, et al. Discovery of 6-({4-[2-(4-tert-butylphenyl)-1H-benzimidazol-4-yl]piperazin-1-yl}methyl)quinoxaline (WAY-207024): an orally active antagonist of the gonadotropin releasing hormone receptor (GnRH-R). J Med Chem. 2009 Apr 9;52(7):2148-52.

Chemical & Physical Properties

[ Molecular Formula ]:
C₃₀H₃₄Cl₂N₆

[ Molecular Weight ]:
549.54

[ Exact Mass ]:
512.24600

[ PSA ]:
60.94000

[ LogP ]:
6.59770

Related Compounds

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