IBZM

Names

[ CAS No. ]:
84226-06-2

[ Name ]:
IBZM

[Synonym ]:
IBZM
(s)-benzamid
N-[[(2S)-1-Ethyl-2-pyrrolidinyl]methyl]-2-hydroxy-3-iodo-6-methoxybenzamide
S-(-)-IBZM
IODOBENZAMIDE,(S)-(-)-3-IODO-2-HYDROXY-6-METHOXY-N[(1-ETHYL-2-PYRROLIDINYL)METHYL]BENZAMIDE
3-iodo-2-hydroxy-6-methoxy-n-((1-ethyl-2-pyrrolidinyl)methyl)benzamide
[123I]-IBZM
(s)-n-(1-ethyl-2-pyrrolidinyl)methyl-2-hydroxy-3-iodo-6-methoxybenzamide
(S)-N-(1-ethylpyrrolidin-2-ylmethyl)-2-hydroxy-3-iodo-6-methoxybenzamide
(S)-(-)-3-iodo-2-hydroxy-6-methoxy-N-[(1-ethyl-2-pyrrolidinyl)methyl]benzamide

Chemical & Physical Properties

[ Density]:
1.51 g/cm3

[ Boiling Point ]:
426.9ºC at 760 mmHg

[ Molecular Formula ]:
C15H21IN2O3

[ Molecular Weight ]:
404.24300

[ Flash Point ]:
212ºC

[ Exact Mass ]:
404.06000

[ PSA ]:
61.80000

[ LogP ]:
2.54830

Toxicological Information

CHEMICAL IDENTIFICATION

RTECS NUMBER :
CV4927050
CHEMICAL NAME :
Benzamide, N-((1-ethyl-2-pyrrolidinyl)methyl)-2-hydroxy-3-iodo-6 -methoxy-, (S)-
CAS REGISTRY NUMBER :
84226-06-2
LAST UPDATED :
199612
DATA ITEMS CITED :
2
MOLECULAR FORMULA :
C15-H21-I-N2-O3
MOLECULAR WEIGHT :
404.28

HEALTH HAZARD DATA

ACUTE TOXICITY DATA

TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Intravenous
SPECIES OBSERVED :
Rodent - rat
DOSE/DURATION :
400 mg/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
REFERENCE :
DCTODJ Drug and Chemical Toxicology. (Marcel Dekker, 270 Madison Ave., New York, NY 10016) V.1- 1977/78- Volume(issue)/page/year: 11,433,1988
TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Intravenous
SPECIES OBSERVED :
Rodent - rabbit
DOSE/DURATION :
50 mg/kg
TOXIC EFFECTS :
Lungs, Thorax, or Respiration - chronic pulmonary edema
REFERENCE :
DCTODJ Drug and Chemical Toxicology. (Marcel Dekker, 270 Madison Ave., New York, NY 10016) V.1- 1977/78- Volume(issue)/page/year: 11,433,1988

Synthetic Route

Precursor & DownStream


Related Compounds