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[Orn5]-URP TFA

Names

[ CAS No. ]:
782485-03-4

[ Name ]:
[Orn5]-URP TFA

Biological Activity

[Description]:

[Orn5]-URP is a potent and selective pure antagonist of Urotensin-II receptor (UT), with an pEC50 of 7.24. [Orn5]-URP displays no agonist activity[1][2].

[Related Catalog]:

Research Areas >> Cardiovascular Disease
Signaling Pathways >> GPCR/G Protein >> Urotensin Receptor

[Target]

pEC50: 7.24[2]


[References]

[1]. Diallo M, et, al. [Orn5]URP acts as a pure antagonist of urotensinergic receptors in rat cortical astrocytes. Peptides. 2008 May; 29(5): 813-9.

[2]. David C, et, al. Structure-activity relationships and structural conformation of a novel urotensin II-related peptide. Peptides. 2004 Oct; 25(10): 1819-30.

Chemical & Physical Properties

[ Molecular Formula ]:
C48H62N10O10S2

[ Molecular Weight ]:
1003.20

[ Storage condition ]:
-20°C

Related Compounds