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San78-130

Names

[ CAS No. ]:
66018-45-9

[ Name ]:
San78-130

Biological Activity

[Description]:

San78-130 is a selective and potent ALK1 inhibitor with an IC50 of 62 nM. San78-130 also inhibits FLT4/VEGFR3, KDR/VEGFR2, MEK2, and FLT3 with IC50s of 114, 162, 186.7, and 188 nM, respectively[1].

[Related Catalog]:

Research Areas >> Cancer

[Target]

ALK1:62 nM (IC50)

FLT4/VEGFR3:114 nM (IC50)

KDR/VEGFR2:162 nM (IC50)

MEK2:186.7 nM (IC50)

FLT3:188 nM (IC50)


[References]

[1]. Cho H, et al. Identification of the First Selective Activin Receptor-Like Kinase 1 Inhibitor, a Reversible Version of L-783277. J Med Chem. 2017 Feb 23;60(4):1495-1508.

Chemical & Physical Properties

[ Molecular Formula ]:
C19H26O7

[ Molecular Weight ]:
366.41

Related Compounds