JNJ-17156516

Names

[ CAS No. ]:
649551-06-4

[ Name ]:
JNJ-17156516

[Synonym ]:
unii-1hxf46y439

Biological Activity

[Description]:

JNJ-17156516 is a你orally active, potent, and selective cholecystokinin (CCK)1-receptor antagonist[1].

[Related Catalog]:

Signaling Pathways >> GPCR/G Protein >> Cholecystokinin Receptor

Research Areas >> Inflammation/Immunology

[References]

[1]. Morton MF, et al. 3-[5-(3,4-Dichloro-phenyl)-1-(4-methoxy-phenyl)-1H-pyrazol-3-yl]-2-m-tolyl-propionate (JNJ-17156516), a novel, potent, and selective cholecystokinin 1 receptor antagonist: in vitro and in vivo pharmacological comparison with dexloxiglumide. J Pharmacol Exp Ther. 2007;323(2):562-569.IF: 3.5 Q2 B2

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₆H₂₂Cl₂N₂O₃

[ Molecular Weight ]:
481.37000

[ Exact Mass ]:
480.10100

[ PSA ]:
64.35000

[ LogP ]:
6.57400