6-Raloxifene-β-D-glucopyranoside

Names

[ Name ]:
6-Raloxifene-β-D-glucopyranoside

Biological Activity

[Description]:

6-Raloxifene-β-D-glucopyranoside, a derivative of Raloxifene, is a benzothiophene glucuronidated at the 6' postion. 6-Raloxifene-β-D-glucopyranoside is a selective and orally active estrogen receptor antagonist. 6-Raloxifene-β-D-glucopyranoside can be used for inhibiting bone loss and resorption, and lowering lipid levels. 6'-Raloxifene-β-D-glucopyranoside, compound Ia, is extracted from patent US5567820A[1].

[Related Catalog]:

Signaling Pathways >> Others >> Estrogen Receptor/ERR

Research Areas >> Metabolic Disease

[Target]

IC50: estrogen receptor[1]

[References]

[1]. Jeffrey A. Dodge, et al. Glucopyranoside benzothiophenes. Patent US5567820A.

Chemical & Physical Properties

[ Molecular Formula ]:
C₃₄H₃₇NO₉S

[ Molecular Weight ]:
635.72

Related Compounds

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