PROTAC PTPN2 degrader-2 TFA

Names

[ CAS No. ]:
2912307-39-0

[ Name ]:
PROTAC PTPN2 degrader-2 TFA

Biological Activity

[Description]:

PROTAC PTPN2 degrader-2 (example 187B) TFA is a potent PTPN2 degrader with potential for studying cancer or metabolic diseases[1].

[Related Catalog]:

Signaling Pathways >> Metabolic Enzyme/Protease >> Phosphatase
Research Areas >> Metabolic Disease
Signaling Pathways >> PROTAC >> PROTAC

[References]

[1]. Protein tyrosine phosphatase targeting ligands.WO2023019166.

Chemical & Physical Properties

[ Molecular Formula ]:
C51H50ClF3N6O13S2

[ Molecular Weight ]:
1111.55