JG-2016

Names

[ CAS No. ]:
2887480-87-5

[ Name ]:
JG-2016

Biological Activity

[Description]:

JG-2016 is a potent inhibitor of histone acetyltransferase 1 (HAT1), with an IC50 of 14.8 μM in the HAT1 acetylation assays[1].

[Related Catalog]:

Research Areas >> Cancer
Signaling Pathways >> Epigenetics >> Histone Acetyltransferase

[References]

[1]. Joshua James GRUBER, et al. Modulators of histone acetyltransferase 1 and methods of treatment thereof. Patent, WO2022272313A1.

Chemical & Physical Properties

[ Molecular Formula ]:
C18H21ClN4O3

[ Molecular Weight ]:
376.84