SN05

Names

[ CAS No. ]:
2768663-51-8

[ Name ]:
SN05

Biological Activity

[Description]:

SN05 is a potent amino acid transport (AAT) inhibitor with Kis of 2.77 μM, 0.73 μM, 0.87 μM, 3.7 μM, 7.25 μM, 7.23 μM and 2.22 μM for human ASCT1, rat ASCT2, human ASCT2, EAAT1, EAAT2, EAAC1 and EAAT5, respectively. SN05 can be used for researching anticancer[1].

[Related Catalog]:

Research Areas >> Cancer
Signaling Pathways >> Others >> Others

[Target]

Ki: 2.77 μM (human ASCT1), 0.73 μM (rat ASCT2), 0.87 μM (human ASCT2), 3.7 μM (EAAT1), 7.25 μM (EAAT2), 7.23 μM (EAAC1), 2.22 μM (EAAT5)[1]


[References]

[1]. Christof GREWER, et al. Inhibitors of amino acid transport. WO2022087630A1

Chemical & Physical Properties

[ Molecular Formula ]:
C18H17NO4

[ Molecular Weight ]:
311.33


Related Compounds

The content on this webpage is sourced from various professional data sources. If you have any questions or concerns regarding the content, please feel free to contact service1@chemsrc.com.