GNE-7883
Names
[ CAS No. ]:
2648450-42-2
[ Name ]:
GNE-7883
Biological Activity
[Description]:
GNE-7883 is a pan-TEAD inhibitor with anti-cell proliferation activity. GNE-7883 overcomes resistance to KRAS G12C inhibitors in multiple preclinical models by inhibiting YAP/TAZ activation. GNE-7883 may be used in the study of YAP/TAZ-dependent cancers[1].
[Related Catalog]:
[Target]
TEAD[1].
[References]
Chemical & Physical Properties
[ Molecular Formula ]:
C28H29FN6O2
[ Molecular Weight ]:
500.57