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Enlicitide chloride

Names

[ CAS No. ]:
2407527-16-4

[ Name ]:
Enlicitide chloride

Biological Activity

[Description]:

Enlicitide chloride is a potent PCSK9 antagonist. Enlicitide chloride can be used for research of cardiovascular disease, e.g. atherosclerosis, hypercholesterolemia, coronary heart disease, metabolic syndrome, acute coronary syndrome, or related cardiovascular disease and cardiometabolic conditions[1][2].

[Related Catalog]:

Signaling Pathways >> Metabolic Enzyme/Protease >> Ser/Thr Protease
Research Areas >> Cardiovascular Disease

[References]

[1]. Ding FX, et al. Preparation of cyclic peptides as PCSK9 antagonist compounds: World Intellectual Property Organization, WO2019246349. 2019-12-26.

[2]. WHO Drug Information-World Health Organization (WHO).

Chemical & Physical Properties

[ Molecular Formula ]:
C82H110ClFN14O15

[ Molecular Weight ]:
1586.29


Related Compounds