AS-1763

Names

[ Name ]:
AS-1763

Biological Activity

[Description]:

AS-1763 is a potent, selective, noncovalent, and orally available inhibitor of Bruton’s tyrosine kinase (IC50 = 0.85 nM).

[Related Catalog]:

Research Areas >> Cancer

Signaling Pathways >> Protein Tyrosine Kinase/RTK >> Btk

[References]

[1]. Kawahata W, et al. Discovery of AS-1763: A Potent, Selective, Noncovalent, and Orally Available Inhibitor of Bruton's Tyrosine Kinase. J Med Chem. 2021 Oct 14;64(19):14129-14141.

Chemical & Physical Properties

[ Molecular Formula ]:
C₃₃H₃₁FN₆O₃

[ Molecular Weight ]:
578.64

Related Compounds

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