DKFZ-251
Names
[ CAS No. ]:
2222059-70-1
[ Name ]:
DKFZ-251
Biological Activity
[Description]:
DKFZ-251 (DKFZ251) is a selective inhibitor of Kallikrein-related peptidase 6 (KLK6) with IC50 of 0.13 uM, demonstrates good selectivity for KLK6 compared to other KLKs; DKFZ-633 exhibits on-target activity in a cellular assay.
[References]
References 1. De Vita E, et al. J Med Chem. 2018 Sep 28. doi: 10.1021/acs.jmedchem.8b01106. View Related Products by Target Other Targets
Chemical & Physical Properties
[ Molecular Formula ]:
C24H24N4O3
[ Molecular Weight ]:
416.481
Related Compounds
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