CARM1 inhibitor 9

Names

[ Name ]:
CARM1 inhibitor 9

Biological Activity

[Description]:

CARM1 inhibitor 9 is a potent, selective inhibitor of arginine methyltransferase 1 (CARM1, PRMT4) with IC50 of 94 nM; displays 20-fold selective for CARM1 over PRMT6 and highly selective over PRMT1, PRMT3, PRMT8 as well as PRMT5 and PRMT7; CARM1 inhibitor 9 is a useful tool for studying the role of CARM1 in health and disease.

[References]

References 1. Kaniskan HÜ, et al. Medchemcomm. 2016 Sep 1;7(9):1793-1796. View Related Products by Target Histone Methyltransferase (HMTase)

Chemical & Physical Properties

[ Molecular Formula ]:
C₁₅H₂₄BrN₃

[ Molecular Weight ]:
326.282

Related Compounds

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