TGR5 agonist 3

Names

[ CAS No. ]:
2148317-51-3

[ Name ]:
TGR5 agonist 3

Biological Activity

[Description]:

TGR5 agonist 3 (compound 8), a Cholic acid derivative, is a selective TGR5 agonist with an EC50 of 5 μM[1].

[Related Catalog]:

Signaling Pathways >> GPCR/G Protein >> GPCR19

Research Areas >> Inflammation/Immunology

[References]

[1]. Emiliano Rosatelli, et al. Chemical exploration of TGR5 functional hot-spots: Synthesis and structure-activity relationships of C7- and C23-Substituted cholic acid derivatives. Eur J Med Chem. 2023 Oct 1:261:115851.

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₈H₄₈O₅

[ Molecular Weight ]:
464.68

Related Compounds

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