tert-butyl 3-{5-chloro-1H-pyrazolo[3,4-b]pyridin-1-yl}azetidine-1-carboxylate

1-{2-Cyclopropylpyrazolo[1,5-a]pyrazin-4-yl}-4-(2-phenylethyl)piperazine

1,3,5-trimethyl-N-{2-[5-(1-methyl-1H-pyrazol-4-yl)thiophen-2-yl]ethyl}-1H-pyrazole-4-sulfonamide

4-(3,5-dimethyl-1H-pyrazol-1-yl)-6-{4-[2-(4-methoxyphenyl)ethyl]piperazin-1-yl}pyrimidine

ethyl 1-[(2-chloro-6-fluorophenyl)methyl]-4-(2,2-dimethoxyethyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazole-3-carboxylate

7-Chloro-2-[4-(cyclopropanesulfonyl)-1,4-diazepan-1-yl]-4-methoxy-1,3-benzothiazole

4-{[1-(2-Fluorobenzenesulfonyl)piperidin-4-yl]methoxy}-3-methylpyridine

4-(1H-pyrazol-1-yl)-6-(4-{pyrazolo[1,5-a]pyrazin-4-yl}piperazin-1-yl)pyrimidine

3-{4-[2-(4-bromophenyl)ethyl]piperazin-1-yl}-6-(1H-pyrazol-1-yl)pyridazine

N-{2-[5-(1-methyl-1H-pyrazol-4-yl)thiophen-2-yl]ethyl}-N'-(1,2-oxazol-3-yl)ethanediamide

4-(4-{2-methylpyrazolo[1,5-a]pyrazin-4-yl}piperazin-1-yl)-6-(1H-pyrazol-1-yl)pyrimidine