BRD-IN-26
Names
[ CAS No. ]:
1915012-19-9
[ Name ]:
BRD-IN-26
Biological Activity
[Description]:
BRD-IN-26 is a potent bromodomain inhibitor that binds the fifth bromodomain of PB1 with a KD of 124 nM, SMARCA2B and SMARCA4 with KD values of 262 and 417 nM, respectively; displays excellent selectivity over other bromodomains.
[References]
References 1. Sutherell CL, et al. J Med Chem. 2016 May 26;59(10):5095-101. View Related Products by Target Bromodomain
Chemical & Physical Properties
[ Molecular Formula ]:
C17H19ClN4O
[ Molecular Weight ]:
330.816