V-9302

Names

[ Name ]:
V-9302

Biological Activity

[Description]:

V-9302 is a competitive antagonist of transmembrane glutamine flux that selectively and potently targets the amino acid transporter ASCT2 with an IC50 of 9.6 μM. V-9302 exhibits anti-tumor activity[1].

[Related Catalog]:

Research Areas >> Cancer

Signaling Pathways >> Others >> Others

[Target]

IC50: 9.6 μM (ASCT2)[1]

[References]

[1]. Schulte ML, et al. Pharmacological blockade of ASCT2-dependent glutamine transport leads to antitumor efficacyin preclinical models. Nat Med. 2018 Feb;24(2):194-202.

Chemical & Physical Properties

[ Molecular Formula ]:
C₃₄H₃₈N₂O₄

[ Molecular Weight ]:
538.68

[ Storage condition ]:
2-8℃

Related Compounds

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