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GSK-8573

Names

[ CAS No. ]:
1693766-04-9

[ Name ]:
GSK-8573

[Synonym ]:
Ethanone, 1-[1-(3-methoxyphenyl)-7-propoxy-3-indolizinyl]-
1-[1-(3-Methoxyphenyl)-7-propoxy-3-indolizinyl]ethanone
GSK-8573

Biological Activity

[Description]:

GSK8573 (compound 23) is an inactive control compound for GSK2801. GSK8573 has binding activity to BRD9 with a Kd value of 1.04 μM and is inactive against BAZ2A/B and other bromodomain familiy[1].

[Related Catalog]:

Research Areas >> Cancer

[Target]

BRD9:1.04 μM (Kd)


[References]

[1]. Chen P, et al. Discovery and Characterization of GSK2801, a Selective Chemical Probe for the Bromodomains BAZ2A and BAZ2B. J Med Chem. 2016 Feb 25;59(4):1410-24.

Chemical & Physical Properties

[ Density]:
1.1±0.1 g/cm3

[ Molecular Formula ]:
C20H21NO3

[ Molecular Weight ]:
323.386

[ Exact Mass ]:
323.152130

[ LogP ]:
4.44

[ Index of Refraction ]:
1.569

[ Storage condition ]:
-20℃

Related Compounds