PDE10A-IN-31
Names
[ CAS No. ]:
1639889-98-7
[ Name ]:
PDE10A-IN-31
Biological Activity
[Description]:
PDE10A-IN-31 is a potent, highly selective PDE10A inhibitor with IC50 of 2 nM for both rPDE10A and hPDE10A; dispalys >2,000-fold selective over PDE1B/2A/3B/4D/5A/7A9A, weak activity on CYP isoforms; displays excellent pharmacokinetic properties.
[References]
References 1. Meegalla SK, et al. Bioorg Med Chem Lett. 2016 Sep 1;26(17):4216-22. View Related Products by Target Phosphodiesterase (PDE)
Chemical & Physical Properties
[ Molecular Formula ]:
C28H23N5O3
[ Molecular Weight ]:
477.524