PDE10A-IN-31

Names

[ Name ]:
PDE10A-IN-31

Biological Activity

[Description]:

PDE10A-IN-31 is a potent, highly selective PDE10A inhibitor with IC50 of 2 nM for both rPDE10A and hPDE10A; dispalys >2,000-fold selective over PDE1B/2A/3B/4D/5A/7A9A, weak activity on CYP isoforms; displays excellent pharmacokinetic properties.

[References]

References 1. Meegalla SK, et al. Bioorg Med Chem Lett. 2016 Sep 1;26(17):4216-22. View Related Products by Target Phosphodiesterase (PDE)

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₈H₂₃N₅O₃

[ Molecular Weight ]:
477.524

Related Compounds

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