RSK2-IN-20

Names

[ Name ]:
RSK2-IN-20

Biological Activity

[Description]:

RSK2-IN-20 is a potent, selective, and durable inhibitpr of RSK2 with IC50 of 47 nM; shows high selectivity over NEK2, PLK1; potently inhibits MSK1 autophosphorylation in cells, and has no significant effect on a panel of 18 additional kinases.

[References]

References 1. Krishnan S, et al. J Am Chem Soc. 2014 Sep 10;136(36):12624-30. View Related Products by Target Ribosomal S6 Kinase (RSK)

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₁H₁₈N₆O₃

[ Molecular Weight ]:
402.414

Related Compounds

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