Usmarapride

Names

[ Name ]:
Usmarapride

[Synonym ]:
Suvn-D4010 Oxalate
1-Isopropyl-3-{5-[1-(3-methoxypropyl)-4-piperidinyl]-1,3,4-oxadiazol-2-yl}-1H-indazole ethanedioate (1:1)
1H-Indazole, 3-[5-[1-(3-methoxypropyl)-4-piperidinyl]-1,3,4-oxadiazol-2-yl]-1-(1-methylethyl)-, ethanedioate (1:1)

Biological Activity

[Description]:

Usmarapride (SUVN-D4010) is a selective 5-HT4 receptor ligand with EC50 value 27.5nM, intended for the symptomatic research of Alzheimer's disease and other disorders of memory and cognition like attention deficient hyperactivity, Parkinson's and schizophrenia[1].

[Related Catalog]:

Research Areas >> Neurological Disease

Signaling Pathways >> GPCR/G Protein >> 5-HT Receptor

Signaling Pathways >> Neuronal Signaling >> 5-HT Receptor

[References]

[1]. Nirogi, Ramakrishna; Mohammed, Abdul Rasheed; Yarlgadda, Suresh; Ravella, Srinivasa Rao; Shinde, Anil Karbhari; Kambhampati, Ramasastri; Roayalley, Praveen Kumar; Jayarajan, Pradeep; Bhyrapuneni, Gopinadh; Patnala, Sriramachandra Murthy; et al. Preparation of heteroaryl compounds as 5-HT4 receptor ligands.WO2013042135A1

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₃H₃₁N₅O₆

[ Molecular Weight ]:
473.52

[ Exact Mass ]:
473.227448

Related Compounds

The content on this webpage is sourced from various professional data sources. If you have any questions or concerns regarding the content, please feel free to contact service1@chemsrc.com.