PR-893

Names

[ Name ]:
PR-893

Biological Activity

[Description]:

A potent, specific immunoproteasome β5 subunit inhibitor with IC50 of 17 nM, 21-fold and 13-fold selectivity for β5 over LMP7 and LMP2 subunits, respecitvely.

[References]

References 1. Parlati F, et al. Blood. 2009 Oct 15;114(16):3439-47. 2. de Bruin G, et al. J Med Chem. 2014 Jul 24;57(14):6197-209. View Related Products by Target Proteasome

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₃H₃₄N₄O₇

[ Molecular Weight ]:
478.546

Related Compounds

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