ERα ligand 1

Names

[ CAS No. ]:
138219-84-8

[ Name ]:
ERα ligand 1

Biological Activity

[Description]:

ERα ligand 1 is an estrogen ligand, which targets estrogen receptor α (ERα). ERα ligand 1 binds to cIAP1 ligand Bestatin via a linker to form PROTACs[1].

[Related Catalog]:

Signaling Pathways >> Others >> Estrogen Receptor/ERR
Research Areas >> Cancer

[References]

[1]. Scheepstra M, et al. Bivalent Ligands for Protein Degradation in Drug Discovery. Comput Struct Biotechnol J. 2019 Jan 25;17:160-176.

Chemical & Physical Properties

[ Molecular Formula ]:
C20H26N2O3

[ Molecular Weight ]:
342.43

Related Compounds