CPI-0610 carboxylic acid

Names

[ Name ]:
CPI-0610 carboxylic acid

Biological Activity

[Description]:

CPI-0610 carboxylic acid is a ligand for target protein for protact. CPI-0610 carboxylic acid is a potent bromodomain and extra-terminal (BET) protein inhibitor in the therapy of multiple myeloma[1].

[Related Catalog]:

Research Areas >> Cancer

Signaling Pathways >> Epigenetics >> Epigenetic Reader Domain

[Target]

BET[1]

[References]

[1]. Albrecht BK, et al. Identification of a Benzoisoxazoloazepine Inhibitor (CPI-0610) of the Bromodomain and Extra-Terminal (BET) Family as a Candidate for Human Clinical Trials. J Med Chem. 2016 Feb 25;59(4):1330-9.

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₀H₁₅ClN₂O₃

[ Molecular Weight ]:
366.80

Related Compounds

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