CTA 056

Names

[ Name ]:
CTA 056

[Synonym ]:
cta-056
cta056

Biological Activity

[Description]:

CTA056 is an ITK (IL-2-inducible T-cell kinase) inhibitor with an IC50 of 0.1 μM. CTA056 selectively targets malignant T cells and modulates oncomirs. CTA056 induces apoptosis and is a potential therapeutic agent for the treatment of T-cell leukemia and lymphoma[1].

[Related Catalog]:

Research Areas >> Cancer

Signaling Pathways >> Protein Tyrosine Kinase/RTK >> Btk

[References]

[1]. Guo W, et al. Molecular characteristics of CTA056, a novel interleukin-2-inducible T-cell kinase inhibitor that selectively targets malignant T cells and modulates oncomirs. Mol Pharmacol. 2012 Nov;82(5):938-47.

Chemical & Physical Properties

[ Molecular Formula ]:
C₃₅H₃₄N₆O

[ Molecular Weight ]:
554.68400

[ Exact Mass ]:
554.27900

[ PSA ]:
79.70000

[ LogP ]:
6.40650

Related Compounds

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