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Sheng Gelieting

Names

[ CAS No. ]:
1152810-23-5

[ Name ]:
Sheng Gelieting

Biological Activity

[Description]:

Sheng Gelieting (CGT-8012) is a dipeptidy peptidase-IV enzyme (DP-IV) inhibitor. Sheng Gelieting has great DP-IV inhibition activity with an IC50 value of 87 nM. Sheng Gelieting can be used for curing or preventing diseases relevant to the dipeptidy peptidase-IV enzyme, such as the diabetes, particularly the II-type diabete[1].

[Related Catalog]:

Research Areas >> Endocrinology
Signaling Pathways >> Metabolic Enzyme/Protease >> Dipeptidyl Peptidase

[Target]

IC50: 87 nM (DP-IV)[1]


[In Vitro]

Sheng Gelieting has great dipeptidy peptidase-IV enzyme (DP-IV) inhibition activity with an IC50 value of 87 nM[1].

[References]

[1]. Qiang Yu, et al. Beta-amino tetrahydropyrazine, tetrahydropyrimidine and tetrahydropyridine used as dipeptidy peptidase inhibitors for curing or preventing diabetes. Patent. CN101899047A.

Chemical & Physical Properties

[ Molecular Formula ]:
C17H16F6N4O

[ Molecular Weight ]:
406.33

Related Compounds