KLK7/ELA2-IN-1

Names

[ CAS No. ]:
1122484-55-2

[ Name ]:
KLK7/ELA2-IN-1

Biological Activity

[Description]:

KLK7/ELA2-IN-1 is a potent kallikrein-related peptidase 7 (KLK7) and epidermal elastase 2 (ELA2) inhibitor with IC50s of 6 nM and 55 nM, respectively (WO2009024527A1, Example 4)[1].

[Related Catalog]:

Research Areas >> Cancer
Signaling Pathways >> Metabolic Enzyme/Protease >> Elastase

[Target]

IC50: 6 nM (KLK7) and 55 nM (ELA2)[1]


[References]

[1]. Philipp Krastel, et al. Cyclic depsipeptides. WO2009024527A1

Chemical & Physical Properties

[ Molecular Formula ]:
C46H72N8O12

[ Molecular Weight ]:
929.11