KLK7/ELA2-IN-1

Names

[ Name ]:
KLK7/ELA2-IN-1

Biological Activity

[Description]:

KLK7/ELA2-IN-1 is a potent kallikrein-related peptidase 7 (KLK7) and epidermal elastase 2 (ELA2) inhibitor with IC50s of 6 nM and 55 nM, respectively (WO2009024527A1, Example 4)[1].

[Related Catalog]:

Research Areas >> Cancer

Signaling Pathways >> Metabolic Enzyme/Protease >> Elastase

[Target]

IC50: 6 nM (KLK7) and 55 nM (ELA2)[1]

[References]

[1]. Philipp Krastel, et al. Cyclic depsipeptides. WO2009024527A1

Chemical & Physical Properties

[ Molecular Formula ]:
C₄₆H₇₂N₈O₁₂

[ Molecular Weight ]:
929.11

KLK7/ELA2-IN-1

Names

Biological Activity

Chemical & Physical Properties

Related Compounds