JNJ-40279486
Names
[ CAS No. ]:
1002351-34-9
[ Name ]:
JNJ-40279486
Biological Activity
[Description]:
JNJ-40279486 is a potent, selective histamine H4 receptor antagonist with Ki of 9.4 nM (hH4), demonstrates acceptable pharmacokinetic profile and efficacy in mouse model of inflammation.
[References]
References 1. Savall BM, et al. Bioorg Med Chem Lett. 2011 Nov 1;21(21):6577-81. View Related Products by Target Histamine Receptor
Chemical & Physical Properties
[ Molecular Formula ]:
C14H15ClN6O
[ Molecular Weight ]:
318.765