Gsk1104252a

Names

[ Name ]:
Gsk1104252a

[Synonym ]:
1-methylethyl 4-({7-[2-fluoro-4-(methylsulfonyl)phenyl]-6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidin-4-yl}oxy)-1 -piperidinecarboxylate

Biological Activity

[Description]:

GSK1104252A is a potent and selective GPR119 agonist. GSK1104252A can be used for type 2 diabetes research[1].

[Related Catalog]:

Signaling Pathways >> GPCR/G Protein >> GPR119

Research Areas >> Metabolic Disease

[References]

[1]. Subba R Katamreddy, et al. Discovery of 6,7-dihydro-5H-pyrrolo[2,3-a]pyrimidines as orally available G protein-coupled receptor 119 agonists. J Med Chem. 2012 Dec 27;55(24):10972-94.

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₂H₂₇FN₄O₅S

[ Molecular Weight ]:
478.53700

[ Exact Mass ]:
478.16900

[ PSA ]:
110.31000

[ LogP ]:
4.18530

Related Compounds

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