Receptor activity and conformational analysis of 5′-halogenated resiniferatoxin analogs as TRPV1 ligands
KS Lim, DW Kang, YS Kim, MS Kim, SG Park…
Index: Bioorganic and Medicinal Chemistry Letters, , vol. 21, # 1 p. 299 - 302
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Citation Number: 5
Abstract
... Bioorganic & Medicinal Chemistry Letters. ... In this Letter, we have investigated the effect of halogenation in the A-region of RTX and of the isosteric 4-amino surrogate in a systematic manner and we describe the synthesis and receptor activity, as well as conformational analysis ...
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[Lim, Kwang Su; Kang, Dong Wook; Kim, Yong Soo; Kim, Myeong Seop; Park, Seul-Gi; Choi, Sun; Pearce, Larry V.; Blumberg, Peter M.; Lee, Jeewoo Bioorganic and Medicinal Chemistry Letters, 2011 , vol. 21, # 1 p. 299 - 302]