Tetrahedron

Synthetic studies on biologically active natural products by a chemicoenzymatic approach: Enantioselective synthesis of C-and N-nucleosides, showdomycin, 6- …

M Ohno, Y Ito, M Arita, T Shibata, K Adachi, H Sawai

Index: Ohno, Masaji; Ito, Yukishige; Arita, Masafumi; Shibata, Tomoyuki; Adachi, Kunitomo; Sawai, Hiroaki Tetrahedron, 1984 , vol. 40, # 1 p. 145 - 152

Full Text: HTML

Citation Number: 67

Abstract

An efficient synthesis of C-and N-nucleosides has been developed in an enantioselective and stereocontrolled manner starting from Diels-Alder adduct of furan and dimethyl acetylenedicarboxylate by chemicoenzymatic strategy. The symmetric unsaturated dimethyl esters 2 and 3 were almost quantitatively hydrolysed with pig liver esterase to yield half- esters 4 and 5 with reasonably high optical yields. Decarboxylative ozonolysis of the chiral ...

Related Articles:

Synthesis of diastereomeric, deoxy and ring-expanded sulfone analogues of aigialomycin D

[Ting, Samuel Z.Y.; Baird, Lynton J.; Dunn, Elyse; Hanna, Reem; Leahy, Dora; Chan, Ariane; Miller, John H.; Teesdale-Spittle, Paul H.; Harvey, Joanne E. Tetrahedron, 2013 , vol. 69, # 49 p. 10581 - 10592]

5'-O-alkyl ethers of N, 2-substituted adenosine derivatives: partial agonists for the adenosine A1 and A3 receptors

[van Tilburg; van der Klein; von Frijtag Drabbe Kuenzel; de Groote; Stannek; Lorenzen; IJzerman Journal of medicinal chemistry, 2001 , vol. 44, # 18 p. 2966 - 2975]

Synthesis of 1, 2, 3-tri-O-acetyl-5-deoxy-D-ribofuranose from D-ribose

[Sairam, Pothukuchi; Puranik, Ramachandra; Sreenivasa Rao, Bhatraju; Veerabhadra Swamy, Ponnapalli; Chandra, Sharad Carbohydrate Research, 2003 , vol. 338, # 4 p. 303 - 306]

The reaction of O-isopropylidene pentodialdo-1, 4-furanoses with lithium diisopropylamide

[Stepowska, Halszka; Zamojski, Aleksander Carbohydrate Research, 1999 , vol. 321, # 1-2 p. 105 - 109]

Efficient tetrahydropyranyl and tetrahydrofuranyl protection/deprotection of alcohols and phenols with Al (OTf) 3 as catalyst

[Williams, D. Bradley G.; Simelane, Sandile B.; Lawton, Michelle; Kinfe, Henok H. Tetrahedron, 2010 , vol. 66, # 25 p. 4573 - 4576]

More Articles...